Phenibut Pure Raw Nootropic Powder CAS 1078-21-3
Product: Phenibut Powder Wholesale
Other Name: 3-Amino-4-phenylbutyric acid hydrochloride
CAS: 060-41-1
MF: C10H14ClNO2
MW: 215.68
MP: 194-201°C
Storage Temp.: Store at RT
Appearance: White cystalline powder.
Physical properties: Phenibut hydrochloride is a white crystalline powder and the taste is very sour. It is readily soluble in water and in alcohol, and the pH of a 2.5% water solution is about 2.3-2.7.
Phenibut Description:
Phenibut is a Russian Nootropic that is most commonly used for boosting mood, treating anxiety and helping to promote healthy sleep. Phenibut is actually derived from GABA, which is a neurotransmitter that is found in the barrier between one’s blood and brain. It was originally discovered in Russia, and people have been using it to treat anxiety in that country since the 1960s. It’s original use was targeted towards astronauts who were dealing with higher levels of stress and anxiety while they were in space for long periods of time. This supplement is often compared to when it comes to its ability to reduce stress, although the strength of Phenibut is not as severe as most pharmaceutical drugs.
Phenibut is a calming, mood lifting, sociability enhancing, and potentially (in low serving sizes) nootropic supplement that acts as a GABA-B agonist to ease stress and support a positive, social mood. The primary benefits of Phenibut use also include pain-reduction, easing muscle tension and stress, and promotion of deep, restful sleep.The recommended serving size of Phenibut is 500 – 2000mg per day, in up to two to three separate servings, depending on the desired effect.
Phenibut Application:
Phenibut is a central depressant and analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA), or a GABA analogue. The addition of a phenyl ring allows phenibut to cross the blood-brain barrier. Phenibut was developed in the Soviet Union in the 1960s, and has since been used there as a pharmaceutical drug to treat a wide range of ailments, including posttraumatic stress disorder, anxiety, depression, asthenia, insomnia, alcoholism, stuttering, and vestibular disorders, and other conditions.
Phenibut is a close structural analogue of GABA, as well as of baclofen (β-(4-chlorophenyl)-GABA), pregabalin (β-isobutyl-GABA), and GABOB (β-hydroxy-GABA). Phenibut is believed to act as a selective GABAB receptor agonist; studies are conflicting as to whether phenibut also acts as a GABAA receptor agonist. More recently, phenibut has been found to act preferentially as a blocker of α2δ subunit-containing voltage-gated calcium channels, similarly to gabapentin and pregabalin. As such, by definition, phenibut is a gabapentinoid.
Phenibut Usage:
1. phenibut is used for post-traumatic stress and vestibular problems.
2. Phenibut uses bodybuilders to reduce fatigue and improve neurological function.
3. Phenibut has been a medical treatment for stress, relieving tension, improving sleep, and acting as other drugs.
4. phenibut induces relaxation and improves psychological functioning.
5. phenibut improves cognition and promotes intelligence and anxiety.
6. phenibut helps fear, anxiety, tension, cognitive impairment, and neurosis in patients with insomnia, depression, and fatigue.
7.Phenibut is a naturally occurring inhibitory neurotransmitter derived from GABA.
Phenibut COA:
| ANALYTICAL ITEMS |
SPECIFICATION |
ANALYTICAL RESULTS |
| Appearance |
White Powder |
White powder |
| Melt Pointing |
194-201°C |
196°C |
| Related substances |
A single impurity≤0.5% |
0.16% |
| Total impurities≤1.0% |
0.37% |
| Loss on drying |
≤0.5% |
0.12% |
| Assay |
>99.0% |
99.5% |
| Conclusion |
Confirms to Enterprise Standard |
Phenibut Benefits:
Phenibut can have a host of benefits when used properly. On the flip-side, using improperly can result in a negative experience that may turn one off from the substance for good. Using the substance for recreational purposes (to get high) will likely lead to a negative experience that can be dangerous and is not recommended.
The benefits of phenibut often relate to calmness and a reduction in anxiety. Phenibut may also help to reduce stress and encourage a better sleep. Finding a “sweet spot” where one can feel the full effects of relaxation without impairing their mental function is how most nootropic users take phenibut. Phenibut should not be used every day and cycled strategically in times of need.
Below and some of the most common benefits experienced with phenibut.
Relaxation
Anxiety reduction
Sleep induction
Reduced stress
Improved mood
Reduces Social Anxiety:
This anxiolytic effect can lead to more rewarding social interactions. There is some limited research supporting enhanced cognitive processing following phenibut consumption, but the primary and supported benefit is anxiolytic.
People that have sought to improve their interactions in social settings have reported better results with the supplement than with alcohol or prescription anxiety medications. Attempted stress and anxiety reduction using traditional tranquilizers often leads to sleepiness and reduced cognitive ability. This undesired side effect isn’t present with phenibut supplementation.
Restores Healthy Sleep Patterns:
People living through depression, anxiety, stressful life events, and hormonal changes, like menopause, often report deteriorating sleep quality. Some have been unsuccessful using melatonin and are unwilling to use pharmaceutical sleep aids. The lack of quality sleep can create an unbroken cycle of impaired cognitive processing, leading to more anxiety, and resulting in even more lost sleep. Phenibut used as an ataractic supplement or sedative can restore helpful, natural sleep patterns, duration, and quality.
We recommend phenibut to persons who are just beginning to experience sleep problems. The ability to fall asleep, remain asleep, and maintain extended periods of healthy, refreshingly deep sleep may be restored quickly with the aid of the supplement. Recapturing healthy sleep patterns early in the destruction process can head off cognitive and emotional problems down the road that may result from the exhaustion.
Phenibut Stacking:
Stacking is the term used when two or more nootropic supplements are taken to derive synergistic benefits through the presence of the other components. This practice has commonly been among nootropic users. An example of this is combining a racetam, like piracetam, with a choline source such as Alpha GPC.
When it comes to phenibut, it is sometimes added to people’s stacks simply to reduce anxiety on days that are extra stressful.
Phenibut Dosage:
The recommended serving size of Phenibut is 500-2000mg per day, in up to two to three separate servings, depending on the desired effect.Phenibut should not be consumed in amounts exceeding 4 grams total per week, and should NEVER be taken in higher amounts on consecutive days due to rapid development of tolerance to the benefits.
Rowe Chen
Sales Manager